Volume 3 No. 3, July 2008

Role of Coenzyme Q10, Metformin and Rosiglitazone in Treatment of Experimental Non Alcoholic Steatohepatitis in Rats
Mohamed A. Abd El- Hamid1, Mahmoud S. Abd El- Halim1, Karima I. El-Desouky2, Heba A. Mahmoud1, Mohamed A. Abdou1

1 Pharmacology & 2Pathology Department, Faculty of Medicine, Tanta University, Egypt

Tanta Med. Sc. J 2008; 3(3):15-29

Article type: Original article

 

Background/Aim: Nonalcoholic fatty liver disease (NAFLD) includes a wide spectrum of liver injury ranging from simple fat accumulation in the hepatocytes (steatosis) without histological or biochemical evidences of inflammation or fibrosis to steatohepatitis with accumulation of fat and necroinflammatory activity. Non-alcoholic steatohepatitis (NASH) is a metabolic liver disorder that is seen in 2-6% of the general population. The aim of the work is to study the effect of each of Coenzyme Q10, metformin and rosiglitazone alone or in certain combination on some parameters of mitochondrial dysfunction in NASH, as mitochondrial ATP& MDA, hepatic TG& FFAs , ALT, AST, fasting blood glucose, serum insulin and HOMA-IR. Materials & Methods: The study was carried out on 80 adult male albino rats weighing 200-250 gram; the animals were classified into 8 groups each group contain10 rats as follow: Group1 (untreated control group) rats were fed on normal diet 12 weeks, Group 2 received high fat diet for 12 weeks, Group 3 received high fat diet and Coenzyme Q10, Group 4 received high fat diet and Metformin, Group 5 received high fat diet and Rosiglitazone, Group 6 received high fat diet and Coenzyme Q10 and Metformin, Group 7 received high fat diet and Coenzyme Q10 and Rosiglitazone, Group 8 received high fat diet and Coenzyme Q10, Rosiglitazone and Metformin. The following parameters were measured: ALT, AST, fasting blood glucose, serum insulin, HOMA- IR, mitochondrial ATP and MDA, hepatic TG and FFAs with histopathological examination. Results: Rosiglitazone induced significant reduction in serum transaminases, fasting blood glucose level, fasting serum insulin, HOMA-IR, mitochondrial MDA, hepatic TG, hepatic FFA. Metformin induced significant reduction in serum transaminases, fasting blood glucose level, fasting serum insulin, HOMA-IR, mitochondrial MDA, hepatic TG, hepatic FFA. Coenzyme Q10 induced significant reduction in serum transaminases, fasting blood glucose level, HOMA-IR, mitochondrial MDA, hepatic FFA with significant increase in mitochondrial ATP. Conclusion: The combination of coenzyme Q10, metformin and rosiglitazone produces additive effect which is very important to decrease hepatic lipid accumulation and insulin resistance which are the two main factors in pathogenesis of NASH.

ICID 870833